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ISSN: 2666-5549

Green polyurethanes from bio-based building blocks: recent advances and applications

Polyurethanes (PUs) are among the most studied, manufactured, and employed polymers thanks to their versatility and wide range of applications. However, their synthesis generally relies on toxic, non-renewable...

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Transaminase catalyzed asymmetric synthesis of active pharmaceutical ingredients

Chiral amine molecules constitute vital components of pharmaceutical ingredients. Recent years have witnessed a growing focus on the efficient synthesis of chiral amines. Transaminases, as catalysts,...

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Carbonylative transformation of aryl halides and strong bonds via cheap metal catalysts and sustainable technologies

The development of catalytic carbonylation reactions has increased considerably. Although many reviews/chapters/books on carbonylation reactions have been published, summaries on cheap metal-catalyzed...

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Recent advances in the syntheses of pyrroles

The pyrrole moiety is an important structural motif in functional materials, natural products, and pharmaceuticals. More and more synthetic strategies toward pyrroles have emerged, where various efficient...

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Ate complexes in organic synthesis: From ate reagents to ate catalysts

The realm of application of organometallic catalysis to organic synthesis has witnessed a transformative shift in recent years, owing much to the evolution of ate complexes from mere reagents to versatile...

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Perspectives on green synthesis and catalysis

Despite their impressive capacity to access diverse functional groups and to synthesize structurally complex molecules, the majority of the organic reactions suffers from harsh conditions, low atom...

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Photocatalytic selective 1,4-oxyimination/diamination across C=C and N=N bonds to access structurally diverse N-N-N triazane derivatives

A highly selective and atom-economical multi-component remote difunctionalization strategy has been successfully developed. This strategy utilizes precise control over the radical properties of bifunctional...

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Advances of Ugi reaction in natural product synthesis

The Ugi multicomponent reaction represents a highly efficient synthetic transformation, wherein all four reactants (isocyanides, amine, aldehyde or ketone and a nucleophile) are combined in one pot...

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Radical azidation as a means of constructing C(sp3)-N3 bonds

The azido group is found in large numbers of natural products, drugs, biochemicals and materials and to date, many elegant and useful methods for the synthesis of organic azides and their transformations...

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Spirooxindoles: Recent report of green synthesis approach

Spirooxindole is a compound with a unique framework and broad bioactivities in medicine. In this study, we have reviewed various approaches or methods in synthesizing spirooxindole derivatives focused...

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Electrochemical generation of nitrogen-centered radicals for organic synthesis

There is a resurgence of interests in organic electrochemistry, which is generally accepted as a green synthetic tool. In this context, many electrochemical methods have been developed in the past decade...

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Organophosphorus catalytic reaction based on reduction of phosphine oxide

The special electronic configuration of phosphorus atoms endows organophosphorus reagents with unique chemical properties, which enable them to be used to catalyze various organic reactions, such as...

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Recent advances in transition-metal-free conversion of aldehydes to ketones

The preparation of functionalized ketones occupies an important position in synthetic organic chemistry because ketones are ubiquitous structural motifs in a broad range of compounds with various applications....

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Flow chemistry in the multi-step synthesis of natural products

The total synthesis of natural products is constantly facing many challenges derived from the complexed chemical structures, the lengthy synthetic routes, the time-consuming workup procedures and the...

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Recent advances in transition-metal-free C–H functionalization of imidazo[1,2-a]pyridines

Imidazo[1,2-a]pyridines are unique nitrogen-containing organic compounds with wide applications in pharmaceuticals, natural products, material science and organometallics. Due to their significant biological...

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1,3-Indanedione: An versatile building block

Indanone-containing compounds are very important components of various natural products, chemical drugs, agrochemicals and functionalized material fields. 1,3-Indanedione is a typical cyclic 1,3-dicarbonyl...

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Synthesis of 5-hydroxymethylfurfural from dehydration of biomass-derived glucose and fructose using supported metal catalysts

The global energy shortage has become more and more serious, which promotes the urgent need to shift to sustainable development. The value-added 5-hydroxymethylfurfural (HMF) can be derived from biomass...

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Photochemical nitrene transfer reactions of iminoiodinanes with sulfoxides

Nitrene, as an important and intriguing versatile synthon, is widely utilized for the formation of diverse nitrogenous skeletons under thermal or photochemical conditions. Typically, the N-sulfonyl...

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Synthesis of tetraarylmethanes: 1897–2022

Tetraarylmethanes (TAMs) contain a carbon atom bound to four aryl groups. They have found diverse applications in chemistry, materials science, chemical biology and medicinal chemistry because of their...

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Synthesis of 1,4-oxathiins via [3+3] annulation of pyridinium 1,4-zwitterionic thiolates with iodonium ylides

A straightforward and valuable approach for the synthesis of 1,4-oxathiins has been developed via [3 ​+ ​3] annulation of pyridinium 1,4-zwitterionic thiolates with iodonium ylides. C–S and C–O bonds...

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Synthesis of indoles, indolines, and carbazoles via palladium-catalyzed C–H activation

The construction of indole, indoline and carbazole heterocycles has been of significant interest in the synthetic community over the last century due to their prevalence in natural products and other...

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Recent advances in visible-light photoredox-catalyzed nitrogen radical cyclization

Visible-light photoredox catalysis is a powerful and attractive strategy for organic molecule activation and new reaction design owing to its environmental-friendly characteristics and unique catalytic...

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Diversification of pharmaceutical molecules via late-stage C(sp2)–H functionalization

C–H late-stage functionalization has gradually become a powerful approach for the rapid optimization of lead compounds’ bioactivity. Significant advances in this field have been achieved in the past...

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Transition-metal-catalyzed transformations of C–N single bonds: Advances in the last five years, challenges and prospects

Nitrogen atom widely exists in many organic molecules and biomacromolecules. Therefore, the formation and transformation of C–N bonds are one of the most attractive topics in organic synthetic chemistry....

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Development of catalyst-free carbon-sulfur bond formation reactions under aqueous media and their applications

Methods for the carbon-sulfur bond formation under catalyst-free, aqueous conditions are extremely useful in organic synthesis and chemical biology. Our laboratory has developed methodologies to construct...

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